Bromadoline powder

Description

Bromadoline powder
Bromadoline powder (U-47931E) is an opioid analgesic selective for the ?-opioid. Buy U47931E Bromadoline powder online with 100% purity.

Product Description
U-47931E (Item No. 20530) is an analytical reference standard that is structurally categorized as an opioid. It has been characterized as a selective µ-opioid receptor agonist, based on the ability of the antagonist ?-funaltrexamine to block U-47931E-mediated decrease in urine output in water-loaded rats. U-47931E has antinociceptive activity comparable to codeine (Item No. ISO60140) in mouse abdominal constriction and rat paw pressure tests.2 This product is intended for research and forensic applications.

Bromadoline maleate
WARNING: This product is for research use only, not for human or veterinary use.

MedKoo CAT#: 328061

CAS#: 81447-81-6 (maleate)

Description: Bromadoline maleate is discontinued (DEA controlled substance). Bromadoline, also known as U-47931E, is an opioid analgesic selective for the ?-opioid receptor. The drug has a potency lying between that of codeine and morphine, being slightly stronger than pentazocine. Bromadoline is related to AH-7921 and U-47700.

Bromadoline maleate is discontinued (DEA controlled substance).
CHEMICAL STRUCTURE
Bromadoline powder
Bromadoline powder

THEORETICAL ANALYSIS
MedKoo Cat#: 328061
Name: Bromadoline maleate
CAS#: 81447-81-6 (maleate)
Chemical Formula: C19H25BrN2O5
Exact Mass: 324.0837
Molecular Weight: 441.322
Elemental Analysis: C, 51.71; H, 5.71; Br, 18.11; N, 6.35; O, 18.13

Related CAS #: 67579-24-2 (free base)

Synonym: Bromadoline; U-47931E; U 47931E; U47931E; U 47,931E; U47,931E; U-47,931E; Bromadoline maleate

IUPAC/Chemical Name: 4-bromo-N-((1R,2R)-2-(dimethylamino)cyclohexyl)benzamide maleate

InChi Key: XHCXKGFNPZETQY-VAYAAYOLSA-N

InChi Code: InChI=1S/C15H21BrN2O.C4H4O4/c1-18(2)14-6-4-3-5-13(14)17-15(19)11-7-9-12(16)10-8-11;5-3(6)1-2-4(7)8/h7-10,13-14H,3-6H2,1-2H3,(H,17,19);1-2H,(H,5,6)(H,7,8)/b;2-1-/t13-,14-;/m1./s1

SMILES Code: O=C(N[C@H]1[C@H](N(C)C)CCCC1)C2=CC=C(Br)C=C2

TECHNICAL DATA
Appearance:Solid powder
Purity:>98% (or refer to the Certificate of Analysis)
Shipping Condition:Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.
Storage Condition:Dry, dark and at 0 – 4 C for short term (days to weeks) or -20 C for long term (months to years).
Solubility:Soluble in DMSO
Shelf Life:>2 years if stored properly
Drug Formulation:This drug may be formulated in DMSO
Stock Solution Storage:0 – 4 C for short term (days to weeks), or -20 C for long term (months).
Harmonized System Code:293490